A Study to Evaluate Pharmacodynamics, Safety, Tolerability and Pharmacokinetics of MT-3995 in Type II Diabetic Nephropathy Subjects With Albuminuria and Moderately Decreased GFR

This study is currently recruiting participants.
Verified March 2013 by Mitsubishi Tanabe Pharma Corporation
Sponsor:
Information provided by (Responsible Party):
Mitsubishi Tanabe Pharma Corporation
ClinicalTrials.gov Identifier:
NCT01756716
First received: December 20, 2012
Last updated: March 14, 2013
Last verified: March 2013
  Purpose

The purpose of this study is to evaluate pharmacodynamics, safety, tolerability and pharmacokinetics of MT-3995 in Type II Diabetic Nephropathy Subjects with Albuminuria and Moderately Decreased GFR


Condition Intervention Phase
Diabetic Nephropathy
Drug: MT-3995 Low
Drug: MT-3995 High
Drug: Placebo
Phase 2

Study Type: Interventional
Study Design: Allocation: Randomized
Endpoint Classification: Safety/Efficacy Study
Intervention Model: Parallel Assignment
Masking: Double Blind (Subject, Investigator)
Primary Purpose: Treatment
Official Title: A Randomised, Double-blind, Placebo-controlled Study to Evaluate the Effect on Urine Albumin-to-Creatinine Ratio (UACR), Pharmacodynamics, Safety, Tolerability and Pharmacokinetics of Multiple Oral Doses of MT-3995 as Add-on Therapy to ACE-I or ARB in Type II Diabetic Nephropathy Subjects With Albuminuria and an eGFR ≥30-<60 mL/Min/1.73m^2

Resource links provided by NLM:


Further study details as provided by Mitsubishi Tanabe Pharma Corporation:

Primary Outcome Measures:
  • Percentage change from baseline in Urine albumin-to-creatinine ratio (UACR) within group. [ Time Frame: up to 8 weeks ] [ Designated as safety issue: No ]
  • Frequency and nature of treatment-emergent adverse events and serious adverse events. [ Time Frame: up to 16 weeks ] [ Designated as safety issue: Yes ]

Secondary Outcome Measures:
  • Percentage change from baseline in UACR compared to placebo [ Time Frame: up to 8 weeks ] [ Designated as safety issue: No ]
  • Change from baseline in Systolic Blood Pressure and Diastolic Blood Pressure within group. [ Time Frame: up to 8 weeks ] [ Designated as safety issue: No ]
  • Plasma concentrations of MT-3995 and its major metabolite [ Time Frame: up to 16 weeks ] [ Designated as safety issue: No ]

Estimated Enrollment: 90
Study Start Date: December 2012
Estimated Study Completion Date: December 2013
Estimated Primary Completion Date: December 2013 (Final data collection date for primary outcome measure)
Arms Assigned Interventions
Experimental: MT-3995 Low group Drug: MT-3995 Low
MT-3995 Low dose for 8 weeks
Experimental: MT-3995 High group Drug: MT-3995 High
MT-3995 High dose for 8 weeks
Placebo Comparator: Placebo group Drug: Placebo
Placebo for 8 weeks

  Eligibility

Ages Eligible for Study:   18 Years to 75 Years
Genders Eligible for Study:   Both
Accepts Healthy Volunteers:   No
Criteria

Inclusion Criteria:

  • Subjects with Type II diabetic nephropathy, who have been treated with angiotensin converting enzyme-inhibitor (ACE-I) or angiotensin II receptor blocker (ARB)
  • Glycosylated haemoglobin (HbA1c) ≤10.5%
  • An estimated glomerular filtration rate (eGFR) ≥30-<60 mL/min/1.73m^2
  • Subject with macroalbuminuria

Exclusion Criteria:

  • History of Type I diabetes, pancreas or β-cell transplantation, or diabetes secondary to pancreatitis or pancreatectomy
  • Serum potassium level <3.5 or >5.0 mmol/L
  • Subjects who had acute kidney injury (AKI) within 3 months prior to baseline or have undergone renal dialysis at any time prior to randomisation
  • Subjects with a history of renal transplant
  • Subjects with clinically significant hypotension
  Contacts and Locations
Please refer to this study by its ClinicalTrials.gov identifier: NCT01756716

Contacts
Contact: Information Desk at Mitsubishi Pharma Europe information@mitsubishi-pharma.eu

Locations
Bulgaria
Investigational site Recruiting
Blagoevgrad, Bulgaria
Investigational site Recruiting
Gabrovo, Bulgaria
Investigational site Recruiting
Plovdiv, Bulgaria
Investigational site Recruiting
Ruse, Bulgaria
Investigational site Recruiting
Sofia, Bulgaria
Investigational site Recruiting
Varna, Bulgaria
Czech Republic
Investigational site Recruiting
Cesky Krumlov, Czech Republic
Investigational site Recruiting
Ostrava, Czech Republic
Investigational site Recruiting
Ostrava-Vitkovice, Czech Republic
Investigational site Recruiting
Slany, Czech Republic
Investigational site Recruiting
Znojmo, Czech Republic
Hungary
Investigational site Recruiting
Baja, Hungary
Investigational site Recruiting
Debrecen, Hungary
Investigational site Recruiting
Eger, Hungary
Investigational site Recruiting
Kistelek, Hungary
Investigational site Recruiting
Komarom, Hungary
Investigational site Recruiting
Pecs, Hungary
Investigational site Recruiting
Szigetvar, Hungary
Investigational site Recruiting
Szikszo, Hungary
Investigational site Recruiting
Zalaegerszeg, Hungary
Romania
Investigational site Recruiting
Bacau, Romania
Investigational site Recruiting
Buzau, Romania
Investigational site Recruiting
Cluj-Napoca, Romania
Investigational site Recruiting
Deva, Romania
Investigational site Recruiting
Isai, Romania
Investigational site Recruiting
Oradea, Romania
Investigational site Recruiting
Targu Mures, Romania
Investigational site Recruiting
Timisoara, Romania
Slovakia
Investigational site Recruiting
Banska Bystrica, Slovakia
Investigational site Recruiting
Bardejov, Slovakia
Investigational site Recruiting
Bratislava, Slovakia
Investigational site Recruiting
Levice, Slovakia
Investigational site Recruiting
Lucenec, Slovakia
Investigational site Recruiting
Martin, Slovakia
Investigational site Recruiting
Nitra, Slovakia
Investigational site Recruiting
Presov, Slovakia
Investigational site Recruiting
Sturovo, Slovakia
Investigational site Recruiting
Zilina, Slovakia
Sponsors and Collaborators
Mitsubishi Tanabe Pharma Corporation
  More Information

No publications provided

Responsible Party: Mitsubishi Tanabe Pharma Corporation
ClinicalTrials.gov Identifier: NCT01756716     History of Changes
Other Study ID Numbers: MT-3995-E07
Study First Received: December 20, 2012
Last Updated: March 14, 2013
Health Authority: Czech Republic: State Institute for Drug Control
Hungary: National Institute of Pharmacy
Bulgaria: Bulgarian Drug Agency
Romania: Ministry of Public Health
Slovakia: State Institute for Drug Control

Keywords provided by Mitsubishi Tanabe Pharma Corporation:
Diabetic Nephropathy

Additional relevant MeSH terms:
Albuminuria
Diabetic Nephropathies
Kidney Diseases
Proteinuria
Urination Disorders
Urologic Diseases
Urological Manifestations
Signs and Symptoms
Diabetes Complications
Diabetes Mellitus
Endocrine System Diseases

ClinicalTrials.gov processed this record on May 19, 2013