A Study of BI 853520 in Patients With Various Types of Advanced or Metastatic Cancer

This study is currently recruiting participants.
Verified May 2013 by Boehringer Ingelheim Pharmaceuticals
Sponsor:
Information provided by (Responsible Party):
Boehringer Ingelheim Pharmaceuticals
ClinicalTrials.gov Identifier:
NCT01335269
First received: April 7, 2011
Last updated: May 15, 2013
Last verified: May 2013
  Purpose

The primary objective of this trial is to determine the safety and tolerability of BI 853520 monotherapy by defining the maximum tolerated dose (MTD) and recommending the dose for further trials in the development of this compound.

Secondary objectives are

  • determination of the pharmacokinetic (PK) profile;
  • exploratory pharmacodynamic analysis; and
  • collection of preliminary data on anti-tumour efficacy.

Condition Intervention Phase
Neoplasms
Drug: BI 853520
Phase 1

Study Type: Interventional
Study Design: Endpoint Classification: Safety/Efficacy Study
Intervention Model: Single Group Assignment
Masking: Open Label
Primary Purpose: Treatment
Official Title: An Open Label Phase I Dose Finding Study of BI 853520 Administered Orally in a Continuous Dosing Schedule in Patients With Various Advanced or Metastatic Non-hematologic Malignancies

Resource links provided by NLM:


Further study details as provided by Boehringer Ingelheim Pharmaceuticals:

Primary Outcome Measures:
  • Determination of the MTD. It will be defined by the occurrence of dose-limiting toxicities (DLT) during the first treatment cycle of each patient in the dose finding phase [ Time Frame: After the first 28 days of treatment ] [ Designated as safety issue: No ]

Secondary Outcome Measures:
  • Pharmacokinetic parameters of BI 853520 will be determined from plasma analyses after a single oral dose and after repeated dosing, at steady state: Cmax and Area Under the Curve [ Time Frame: During first 28 days of treatment ] [ Designated as safety issue: No ]
  • Pharmacodynamic assessment: pPTK2 modulation pre- and post treatment in skin or tumor [ Time Frame: During the first 28 days of treatment ] [ Designated as safety issue: No ]
  • Exploratory evaluation of efficacy (e.g. objective response rate, disease control rate, duration of disease control, tumor shrinkage) [ Time Frame: Every 8 weeks until end of study participation ] [ Designated as safety issue: No ]

Estimated Enrollment: 90
Study Start Date: July 2011
Estimated Study Completion Date: August 2014
Estimated Primary Completion Date: August 2014 (Final data collection date for primary outcome measure)
Arms Assigned Interventions
Experimental: Treatment arm
BI 853520 once daily in a dose escalation schedule
Drug: BI 853520
BI 853520 once daily in a dose escalation schedule

  Eligibility

Ages Eligible for Study:   18 Years and older
Genders Eligible for Study:   Both
Accepts Healthy Volunteers:   No
Criteria

Inclusion criteria:

  • Patients with a confirmed diagnosis of advanced, measurable or evaluable, non-resectable and/or metastatic non-hematologic malignancy, which has shown to be progressive in the last 6 months
  • Patients who have failed conventional treatment or for whom no therapy of proven efficacy exists or who are not amenable to established treatment options
  • Recovery from reversible toxicities (alopecia excluded) of prior anti-cancer therapies (Common Terminology Criteria for Adverse Events grade <2)
  • Age >= 18 years
  • Written informed consent in accordance with International Conference on Harmonisation/Good Clinical Practice (ICH/GCP) and local legislation
  • Eastern Cooperative Oncology Group (ECOG), performance score 0-1

Exclusion criteria:

  • Serious concomitant non-oncological disease/illness
  • Active/symptomatic brain metastases
  • Second malignancy
  • Pregnancy or breastfeeding
  • Women or men who are sexually active and unwilling to use a medically acceptable method of contraception.
  • Treatment with cytotoxic anti-cancer-therapies or investigational drugs within four weeks of the first treatment with the study medication
  Contacts and Locations
Please refer to this study by its ClinicalTrials.gov identifier: NCT01335269

Contacts
Contact: Boehringer Ingelheim Call Center 1-800-243-0127 clintriage.rdg@boehringer-ingelheim.com

Locations
Canada, Ontario
1300.2.1002 Boehringer Ingelheim Investigational Site Not yet recruiting
Hamilton, Ontario, Canada
1300.2.1001 Boehringer Ingelheim Investigational Site Recruiting
Toronto, Ontario, Canada
Netherlands
1300.2.31001 Boehringer Ingelheim Investigational Site Recruiting
Rotterdam, Netherlands
Sponsors and Collaborators
Boehringer Ingelheim Pharmaceuticals
Investigators
Study Chair: Boehringer Ingelheim Boehringer Ingelheim Pharmaceuticals
  More Information

No publications provided

Responsible Party: Boehringer Ingelheim Pharmaceuticals
ClinicalTrials.gov Identifier: NCT01335269     History of Changes
Other Study ID Numbers: 1300.2, 2010-024609-10
Study First Received: April 7, 2011
Last Updated: May 15, 2013
Health Authority: Canada: Health Canada
Netherlands:

Additional relevant MeSH terms:
Neoplasms

ClinicalTrials.gov processed this record on May 23, 2013